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CAS No. : 54784-44-0
MCE 国际站:[D-Phe2,D-Ala6]-LH-RH
产品活性:[D-Phe2,D-Ala6]-LH-RH 是一种有效的 LH-RH 拮抗剂。[D-Phe2,D-Ala6]-LH-RH 具有抗 LH/FSH-RH 和抗排卵活性。
研究领域:Others
作用靶点:Others
In Vivo: [D-Phe2,D-Ala6]-LH-RH inhibits the LH and FSH release induced by LH-RH in immature male rats.
[D-Phe2,D-Ala6]-LH-RH (1 mg/rat, SC) shows marked antiovulatory and contraceptive activity.[D-Phe2,D-Ala6]-LH-RH (0.625, 1.25, 2.5 mg/kg; s.c.; single dose; sacrificed 30 minutes) results a dose-dependent increase in stalk-median eminence (SME)-LHRH activity and decreases plasma LHRH activity as well in rats with hypophysectomized (hypox) at 25 days old.
[D-Phe2,D-Ala6]-LH-RH (25 mg/kg; s.c.; single dsoe) is effective in blocking the ovulation normally induced by LRH alone.
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