Biological Activity
SYM 2081 is a potent and highly selective kainate receptor agonist, with an IC50for inhibition of [3H]-kainate binding of 35 nM and almost 3,000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively. Also selectively inhibits the cloned excitatory amino acid transporter EAAT2 at higher concentrations.
Technical Data
M.Wt:
161.16
Formula:
C6H11NO4
Solubility:
Soluble to 50 mM in water
Purity:
≥97%
Storage:
Store at RT
CAS No:
31137-74-3
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Catalog # | Availability | Size / Price | |
---|---|---|---|
0903/10 | Contact your distributor for availability. | 10 mg |